Cyclic mimetics of kinase-inhibitory region of Suppressors of Cytokine Signaling 1: Progress toward novel anti-inflammatory therapeutics
Sara La Manna, Laura Lopez‐Sanz, Susana Bernal, Sara Fortuna, Flavia Anna Mercurio, Marilisa Leone, Carmen Gómez‐Guerrero, Daniela Marasco
Topics & Concepts
ChemistrySuppressor of cytokine signaling 1Tyrosine phosphorylationPhosphorylationProinflammatory cytokineCytokinePeptidomimeticSTAT1Biological activityBiochemistrySignal transductionCell biologyInflammationGeneSuppressorBiologyPeptideImmunologyIn vitroCytokine Signaling Pathways and Interactionsinterferon and immune responsesPharmacological Effects of Natural Compounds