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Dual inhibitors of <i>Pseudomonas aeruginosa</i> virulence factors LecA and LasB

Olga Metelkina, Jelena Konstantinović, Andreas Klein, Roya Shafiei, Mario A. Fares, Alaa Alhayek, Samir Yahiaoui, Walid A. M. Elgaher, Jörg Haupenthal, Alexander Titz, Anna K. H. Hirsch

2024Chemical Science14 citationsDOIOpen Access PDF

Abstract

Dual inhibitors of two key virulence factors of Pseudomonas aeruginosa , the lectin LecA and the protease LasB, open up an opportunity in the current antimicrobial-resistance crisis.

Topics & Concepts

Pseudomonas aeruginosaVirulenceMicrobiologyVirulence factorDual (grammatical number)Antibiotic resistanceBiologyBacteriaAntibioticsBiochemistryGeneticsGeneLiteratureArtBacterial biofilms and quorum sensingAntimicrobial Peptides and ActivitiesBiochemical and Structural Characterization
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