Discovery of a potent dual inhibitor of wild-type and mutant respiratory syncytial virus fusion proteins through the modulation of atropisomer interconversion properties
Toru Yamaguchi-Sasaki, Takanori Kawaguchi, Atsushi Okada, Seiken Tokura, Nozomi Tanaka-Yamamoto, Tomoki Takeuchi, Yuya Ogata, Ryo Takahashi, Risa Kurimoto-Tsuruta, Tomokazu Tamaoki, Yutaka Sugaya, Tomoko Abe-Kumasaka, Kaho Arikawa, Ippei Yoshida, Hiroyuki Sugiyama, Kosuke Kanuma, Mitsukane Yoshinaga
Topics & Concepts
AtropisomerChemistryLinkerMoietyPyrimidineMutantStereochemistryFusion proteinWild typeBiochemistryRecombinant DNAGeneComputer scienceOperating systemRespiratory viral infections researchPneumonia and Respiratory InfectionsInfluenza Virus Research Studies