Molecular basis for ligand activation of the human KCNQ2 channel
Xiaoxiao Li, Qiansen Zhang, Peipei Guo, Jie Fu, Lianghe Mei, Dashuai Lv, Jiangqin Wang, Dongwu Lai, Sheng Ye, Huaiyu Yang, Jiangtao Guo
Topics & Concepts
Allosteric regulationActivator (genetics)Drug discoveryPotassium channelChemistryLigand (biochemistry)BiophysicsStructural biologyNeuroscienceBiochemistryBiologyReceptorIon channel regulation and functionCardiac electrophysiology and arrhythmiasNeuroscience and Neural Engineering