A2A Adenosine Receptor Partial Agonism Related to Structural Rearrangements in an Activation Microswitch
Matthew T. Eddy, Bryan Martín, Kurt Wüthrich
Topics & Concepts
Partial agonistAgonistG protein-coupled receptorIntracellularChemistryReceptorAgonismAdenosine receptorSignal transductionAdenosineStereochemistryBiophysicsBiochemistryBiologyPoliticsPolitical scienceLawReceptor Mechanisms and SignalingAdenosine and Purinergic SignalingNeuropeptides and Animal Physiology