Litcius/Paper detail

Evolution in non-peptide α-helix mimetics on the road to effective protein-protein interaction modulators

Sergio Algar, Mercedes Martín‐Martínez, Rosario González‐Muñiz

2020European Journal of Medicinal Chemistry24 citationsDOIOpen Access PDF

Topics & Concepts

PeptidomimeticChemistrySmall moleculeHelix (gastropod)InteractomePeptideProtein–protein interactionPharmacophoreDrug discoveryAmino acidSide chainMoleculeCombinatorial chemistryStereochemistryComputational biologyBiochemistryPolymerEcologyOrganic chemistryGeneSnailBiologyChemical Synthesis and AnalysisClick Chemistry and ApplicationsUbiquitin and proteasome pathways
Evolution in non-peptide α-helix mimetics on the road to effective protein-protein interaction modulators | Litcius