Introducing a pyrazolopyrimidine as a multi-tyrosine kinase inhibitor, using multi-QSAR and docking methods
Asrin Bahmani, Hamid Tanzadehpanah, Neda Hosseinpour Moghadam, Massoud Saidijam
Topics & Concepts
Quantitative structure–activity relationshipDocking (animal)RegorafenibComputational biologyChemistryDrug discoveryReceptor tyrosine kinaseBinding siteStereochemistryBiologyKinaseBiochemistryCancerColorectal cancerGeneticsMedicineNursingSynthesis and biological activityComputational Drug Discovery MethodsHER2/EGFR in Cancer Research