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Photocatalyst-Free, Visible-Light-Mediated C(sp<sup>3</sup>)–H Arylation of Amides via a Solvent-Caged EDA Complex

Jaspreet Kaur, Ahmed Shahin, Joshua P. Barham

2021Organic Letters45 citationsDOIOpen Access PDF

Abstract

A photocatalyst-free and mild visible light photochemical procedure for C(sp3)–H arylation of amides is described. The reaction proceeds via an electron donor–acceptor (EDA) complex between an electron-rich arene substrate and electron-poor persulfate oxidant. C(sp3)–H arylation of the amide occurs selectively with the most electron-rich arene of the substrate. Mechanistic studies corroborate the reaction taking place in a solvent cage holding components in a close proximity.

Topics & Concepts

ChemistryPersulfateSubstrate (aquarium)PhotochemistryElectron acceptorAmidePhotocatalysisVisible spectrumSolventElectron donorCatalysisOrganic chemistryOceanographyOptoelectronicsPhysicsGeologyRadical Photochemical ReactionsSulfur-Based Synthesis TechniquesCatalytic C–H Functionalization Methods