Probing biased activation of mu-opioid receptor by the biased agonist PZM21 using all atom molecular dynamics simulation
Siyan Liao, Kai Tan, Cecilia Floyd, Daegun Bong, Michael James Pino, Chun Wu
Topics & Concepts
G protein-coupled receptorIntracellularMolecular dynamicsAgonistChemistryBiophysicsμ-opioid receptorOpioid receptorReceptorG proteinHeterotrimeric G proteinOpioidStereochemistryBiologyBiochemistryComputational chemistryReceptor Mechanisms and SignalingNeuropeptides and Animal PhysiologyComputational Drug Discovery Methods