Medicinal chemistry strategies targeting PRMT5 for cancer therapy
Siyu Fu, Qinwen Zheng, Dan Zhang, Congcong Lin, Liang Ouyang, Jifa Zhang, Lei Chen
Topics & Concepts
Protein arginine methyltransferase 5ChemistryMethyltransferaseArginineDownregulation and upregulationCancer therapyCancer researchCancerPharmacologyDrug developmentDrugBiochemistryAmino acidMedicineMethylationInternal medicineGeneCancer-related gene regulationEpigenetics and DNA Methylation