The development of Coronavirus 3C-Like protease (3CLpro) inhibitors from 2010 to 2020
Yuzhi Liu, Chengyuan Liang, Liang Xin, Xiaodong Ren, Lei Tian, Xingke Ju, Li Han, Yongbo Wang, Qianqian Zhao, Hong Liu, Wenqiang Cao, Xiaolin Xie, Dezhu Zhang, Yu Wang, Yanlin Jian
Topics & Concepts
ChemistryPeptidomimeticStereochemistryCoronavirusProteaseSmall moleculeCovalent bondHydrogen bondCombinatorial chemistryEnzymeMoleculeCoronavirus disease 2019 (COVID-19)BiochemistryOrganic chemistryPathologyPeptideDiseaseMedicineInfectious disease (medical specialty)Protein Degradation and InhibitorsPeptidase Inhibition and AnalysisCancer therapeutics and mechanisms