Litcius/Paper detail

De novo design of tyrosine and serine kinase-driven protein switches

Nicholas B. Woodall, Zara Y. Weinberg, Jesslyn Park, Florian Büsch, Richard S. Johnson, Mikayla J. Feldbauer, Michael Murphy, Maggie Ahlrichs, Issa Yousif, Michael J. MacCoss, Vicki H. Wysocki, Hana El‐Samad, David Baker

2021Nature Structural & Molecular Biology34 citationsDOIOpen Access PDF

Topics & Concepts

SerineProtein-Tyrosine KinasesCell biologyTyrosineTyrosine kinaseChemistryReceptor tyrosine kinaseBiochemistryBiologyKinaseSignal transductionPhosphorylationUbiquitin and proteasome pathwaysProtein Kinase Regulation and GTPase SignalingComputational Drug Discovery Methods