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Synthesis of New Bioactive Indolyl-1,2,4-Triazole Hybrids As Dual Inhibitors for EGFR/PARP-1 Targeting Breast and Liver Cancer Cells

Mohamed F. Youssef, Mohamed S. Nafie, Eid E. Salama, Ahmed T. A. Boraei, Emad M. Gad

2022ACS Omega29 citationsDOIOpen Access PDF

Abstract

may serve as a promising anticancer activity through dual PARP-1/EGFR target inhibition.

Topics & Concepts

ChemistryCytotoxicityCancer cellMTT assayApoptosisTriazoleCancer researchCancerBiochemistryIn vitroBiologyOrganic chemistryGeneticsSynthesis and biological activityClick Chemistry and ApplicationsCancer therapeutics and mechanisms
Synthesis of New Bioactive Indolyl-1,2,4-Triazole Hybrids As Dual Inhibitors for EGFR/PARP-1 Targeting Breast and Liver Cancer Cells | Litcius