In silico docking and ADME study of deketene curcumin derivatives (DKC) as an aromatase inhibitor or antagonist to the estrogen-alpha positive receptor (Erα+): potent application of breast cancer
Vraj Shah, Jaydip Bhaliya, Gautam M. Patel
Topics & Concepts
AromataseBreast cancerFulvestrantEstrogen receptorEstrogen receptor alphaChemistryADMEPharmacologyTamoxifenEstrogenSelective estrogen receptor modulatorCancerCancer researchDrugInternal medicineMedicineEstrogen and related hormone effectsCurcumin's Biomedical ApplicationsAdvanced Breast Cancer Therapies