Identification of novel 1,3-diaryl-1,2,4-triazole-capped histone deacetylase 6 inhibitors with potential anti-gastric cancer activity
Xinhui Zhang, Huiqin Kang, Yuanyuan Tao, Yihan Li, Junru Zhao, Ya-Gao, Liying Ma, Hong‐Min Liu
Topics & Concepts
HDAC6ChemistryAcetylationHistone deacetylaseHDAC1CancerChemical libraryCancer cellCancer researchHistonePharmacologyBiochemistryBiologySmall moleculeMedicineInternal medicineGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsPeptidase Inhibition and Analysis