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Covalent inhibition of NSD1 histone methyltransferase

Huang Huang, Christina A. Howard, Sergei Zari, Hyo Je Cho, Shirish Shukla, Hao Li, Juliano Ndoj, Paula Gónzález-Alonso, Caroline Nikolaidis, Joshua M. Abbott, David Rogawski, Mykhaylo A. Potopnyk, Katarzyna Kempińska, Hongzhi Miao, Trupta Purohit, Andrew J. Henderson, Anna K. Mapp, Maria Luisa Sulis, Adolfo A. Ferrando, Jolanta Grembecka, Tomasz Cierpicki

2020Nature Chemical Biology87 citationsDOIOpen Access PDF

Topics & Concepts

MethyltransferaseHistone methyltransferaseHistoneChemistryCovalent bondComputational biologyBiochemistryCell biologyBiologyMethylationGeneOrganic chemistryEpigenetics and DNA MethylationCancer-related gene regulationRNA modifications and cancer
Covalent inhibition of NSD1 histone methyltransferase | Litcius