Targeted degradation of anaplastic lymphoma kinase by gold nanoparticle-based multi-headed proteolysis targeting chimeras
Yingming Wang, Lingfei Han, Fulei Liu, Fubai Yang, Xueyang Jiang, Haopeng Sun, Feng Feng, Jingwei Xue, Wenyuan Liu
Topics & Concepts
Ubiquitin ligaseAnaplastic lymphoma kinaseCeritinibFusion proteinChemistryCereblonUbiquitinKinaseProtein degradationCancer researchBiochemistryBiologyMedicineLung cancerRecombinant DNAMalignant pleural effusionGeneInternal medicineProtein Degradation and InhibitorsPeptidase Inhibition and AnalysisMultiple Myeloma Research and Treatments