Anticancer activity of hydrazones in the last quinquennial period: A special emphasis on various enzyme targets and SAR
Shyama Charan, Naazneen Maksud, Amisha Gupta, Sonia Devi, Mohammad Mahtab Alam, Mymoona Akhter, Sharba Tasneem, Darakhshan Parveen, Ahasan, Mohammad Shaquiquzzaman
Topics & Concepts
ChemistryHydrazoneEnzymeCombinatorial chemistryStructure–activity relationshipStereochemistryAnticancer drugComputational biologyDrugBiochemistryArylLead compoundActive siteFlexibility (engineering)Drug discoveryDocking (animal)Chemical synthesisPharmacologyEnzyme inhibitionMechanism of actionEnzyme assayCancer cellBiological activityRational designTyrosineEnzyme inhibitorEnzyme function and inhibitionSynthesis and biological activityChemotherapy-induced cardiotoxicity and mitigation