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Bioanalytical method development and validation for the quantitation of larotrectinib in human plasma: Application to pharmacokinetics in healthy rabbits

Shankar Cheruku, Bhikshapathi Darna, Viswaja Medipalli, Arjuna Rao Nekkalapudi, Rubesh Kumar Sadasivam

2023Journal of Applied Pharmaceutical Science10 citationsDOIOpen Access PDF

Abstract

QSAR, Molecular Docking and Dynamics Studies of Pyrrolo[2,3-b]Pyridine Derivatives as Bruton’s Tyrosine Kinase InhibitorsRuslin, Nirwana, Muhammad Arba, Mukhsar, Daryono Hadi Tjahjono

Topics & Concepts

BioanalysisPharmacokineticsPharmacologyPyridineChemistryHuman plasmaDocking (animal)Tyrosine kinaseStereochemistryComputational biologyChromatographyBiochemistryMedicineBiologyMedicinal chemistrySignal transductionNursingPI3K/AKT/mTOR signaling in cancerChronic Lymphocytic Leukemia ResearchPancreatic and Hepatic Oncology Research
Bioanalytical method development and validation for the quantitation of larotrectinib in human plasma: Application to pharmacokinetics in healthy rabbits | Litcius