Cryo-EM structures of inactive and active GABAB receptor
Chunyou Mao, Cangsong Shen, Chuntao Li, Dandan Shen, Chanjuan Xu, Shenglan Zhang, Rui Zhou, Qingya Shen, Li-Nan Chen, Zhinong Jiang, Jianfeng Liu, Yan Zhang
Topics & Concepts
Allosteric regulationGABAB receptorTransmembrane domainBiophysicsAllosteric modulatorG protein-coupled receptorChemistryProtein subunitAgonistHelix (gastropod)ReceptorBiologyBiochemistrySnailGeneEcologyReceptor Mechanisms and SignalingNeuroscience and Neuropharmacology ResearchIon channel regulation and function