Discovery of 4-hydroxyl pyrazole derivatives as potent ferroptosis inhibitors
Danzhi Ying, Xin Shen, Shuqi Wang, Junyi Chen, Zhenying Wu, Wenteng Chen, Fudi Wang, Junxia Min, Yongping Yu
Topics & Concepts
PyrazoleChemistryProgrammed cell deathEC50Lead compoundPharmacologyIC50Cell cultureIn vitroStereochemistryBiochemistryApoptosisBiologyGeneticsFerroptosis and cancer prognosisCancer, Lipids, and MetabolismRNA modifications and cancer