Litcius/Paper detail

Nonclinical Pharmacokinetics and Absorption, Distribution, Metabolism, and Excretion of Givosiran, the First Approved N-Acetylgalactosamine–Conjugated RNA Interference Therapeutic

Jing Li, Ju Liu, Xuemei Zhang, Valerie A. Clausen, Chris Tran, Michael Arciprete, Qianfan Wang, Carrie Rocca, Lihua Guan, Guodong Zhang, Diana Najarian, Yuanxin Xu, Pete Smith, Jing‐Tao Wu, Saeho Chong

2021Drug Metabolism and Disposition43 citationsDOIOpen Access PDF

Topics & Concepts

PharmacokineticsPharmacologyADMEChemistryCytochrome P450MetabolismExcretionDrug metabolismMetaboliteIsozymeRenal physiologyBiochemistryBiologyEnzymeRenal functionPorphyrin Metabolism and DisordersHeme Oxygenase-1 and Carbon MonoxidePorphyrin and Phthalocyanine Chemistry