Identification of an allosteric hotspot for additive activation of PPARγ in antidiabetic effects
Feng Li, Shaoyong Lu, Zhen Zheng, Ying‐Yi Chen, Yuanyuan Zhao, Kun Song, Hongjuan Xue, Lihua Jin, Yong Li, Yong Li, Cheng Huang, Yiming Li, Yiming Li, Jian Zhang
Topics & Concepts
Allosteric regulationRosiglitazonePharmacologyGlucose homeostasisPeroxisome proliferator-activated receptorChemistryDruggabilityMedicineReceptorBiochemistryDiabetes mellitusEndocrinologyInsulin resistanceGenePeroxisome Proliferator-Activated ReceptorsNF-κB Signaling PathwaysBioactive natural compounds