Design, synthesis, and biological activity evaluation of 2-(benzo[b]thiophen-2-yl)-4-phenyl-4,5-dihydrooxazole derivatives as broad-spectrum antifungal agents
Liyu Zhao, Yin Sun, Wenbo Yin, Linfeng Tian, Nannan Sun, Yang Zheng, Chu Zhang, Shizhen Zhao, Xin Su, Dongmei Zhao, Maosheng Cheng
Topics & Concepts
Cryptococcus neoformansChemistryAspergillus fumigatusCandida albicansAntifungalCYP3A4StereochemistryBroad spectrumPharmacokineticsMinimum inhibitory concentrationIn vitroBiological activityChemical synthesisPharmacologyMetabolismCytochrome P450BiochemistryCombinatorial chemistryMicrobiologyMedicineBiologySynthesis and Biological EvaluationSynthesis and biological activityCancer therapeutics and mechanisms