Inhibiting CDK6 Activity by Quercetin Is an Attractive Strategy for Cancer Therapy
Mohd Yousuf, Parvez Κhan, Anas Shamsi, Mohd Shahbaaz, Gulam Mustafa Hasan, Qazi Mohd Rizwanul Haque, Alan Christoffels, Asimul Islam, Md. Imtaiyaz Hassan
Abstract
studies highlight the significance of quercetin for the development of anticancer leads in terms of CDK6 inhibitors.
Topics & Concepts
QuercetinIsothermal titration calorimetryChemistryCyclin-dependent kinase 6BiochemistryIn silicoPharmacologyApoptosisCell cycleBiologyCyclin D1AntioxidantGeneCancer-related Molecular PathwaysComputational Drug Discovery MethodsCancer, Lipids, and Metabolism