Novel fluoroquinolone hybrids as dual DNA gyrase and urease inhibitors with potential antibacterial activity: Design, synthesis, and biological evaluation
Salah A. Abdel‐Aziz, Katarina Cirnski, Jennifer Herrmann, Mohamed A. A. Abdel‐Aal, Bahaa G. M. Youssif, Ola I. A. Salem
Topics & Concepts
ChemistryNorfloxacinDNA gyraseUreaseCiprofloxacinAntibacterial activityMinimum inhibitory concentrationEscherichia coliIC50BiochemistryBacteriaEnzymeAntibioticsIn vitroBiologyGeneGeneticsCancer therapeutics and mechanismsAntibiotic Resistance in BacteriaPneumocystis jirovecii pneumonia detection and treatment