Novel tacrine-based acetylcholinesterase inhibitors as potential agents for the treatment of Alzheimer’s disease: Quinolotacrine hybrids
Mehrdad Sadafi Kohnehshahri, Gholamabbas Chehardoli, Masoomeh Bahiraei, Tahmineh Akbarzadeh, Akram Ranjbar, Arezoo Rastegari, Zahra Najafi
Topics & Concepts
ButyrylcholinesteraseAcetylcholinesteraseTacrineChemistryCholinesteraseAchéIC50StereochemistryADMEDocking (animal)EnzymePharmacologyBiochemistryIn vitroBiologyMedicineNursingCholinesterase and Neurodegenerative DiseasesNicotinic Acetylcholine Receptors StudyChemical synthesis and alkaloids