Computational approaches for the design of novel dopamine D2 and serotonin 5-HT2A receptor dual antagonist towards schizophrenia
Akash Rathore, Vivek Asati, Mitali Mishra, Ratnesh Das, Varsha Kashaw, Sushil K. Kashaw
Topics & Concepts
ChemistryQuantitative structure–activity relationshipPharmacophoreStereochemistryDopamine receptor D2PiperazineDocking (animal)PiperidineProtein Data Bank (RCSB PDB)ADMEReceptorBiochemistryOrganic chemistryMedicineIn vitroNursingComputational Drug Discovery MethodsReceptor Mechanisms and SignalingPharmacological Receptor Mechanisms and Effects