Iodoquinazoline-derived VEGFR-2 and EGFRT790M dual inhibitors: Design, synthesis, molecular docking and anticancer evaluations
Abeer A. Mohamed, Sanadelaslam S. A. El‐Hddad, Ahmed K. B. Aljohani, Fathalla Khedr, Omar M. Alatawi, Doaa E. Keshek, Sahar Ahmed, Marwa Alsulaimany, Sara A. Almadani, Khaled El‐Adl, Noura S. Hanafy
Topics & Concepts
ChemistryCytotoxicityIC50MTT assayDocking (animal)StereochemistryA549 cellVero cellCell cultureCytotoxic T cellIn vitroPharmacologyBiochemistryBiologyNursingMedicineGeneticsToxin Mechanisms and ImmunotoxinsHER2/EGFR in Cancer ResearchQuinazolinone synthesis and applications