In Vitro and Cellular Probes to Study PARP Enzyme Target Engagement
Tim J. Wigle, Danielle J. Blackwell, Laurie B. Schenkel, Yue Ren, W. David Church, Hetvi J. Desai, Kerren K. Swinger, Andrew G. Santospago, Christina R. Majer, Alvin Lu, Mario Niepel, Nicholas R. Perl, Melissa M. Vasbinder, Heike Keilhack, Kevin W. Kuntz
Topics & Concepts
Poly ADP ribose polymeraseNAD+ kinaseEnzymeBiochemistryPolymerasePARP inhibitorIn vitroNicotinamide adenine dinucleotideIn vitro toxicologyChemistryRiboseNicotinamideBiologyMolecular biologyPARP inhibition in cancer therapyIntegrated Circuits and Semiconductor Failure AnalysisElectrostatic Discharge in Electronics