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SQR mediates therapeutic effects of H <sub>2</sub> S by targeting mitochondrial electron transport to induce mitochondrial uncoupling

Jia Jia, Zichuang Wang, Minjie Zhang, Caiyun Huang, Yanmei Song, XU Fu-you, Jingyu Zhang, Jie Li, Meijun He, Yuyao Li, Gui‐Zhen Ao, Hong Chengjiao, Yongjun Cao, Y. Eugene Chin, Zichun Hua, Jian Cheng

2020Science Advances90 citationsDOIOpen Access PDF

Abstract

S signaling and therapeutic effects by targeting mitochondrial electron transport to induce mitochondrial uncoupling. Moreover, SQR is a previously unrecognized target for developing non-protonophore uncouplers with broad clinical implications.

Topics & Concepts

AMPKMitochondrionCell biologyElectron transport chainUncoupling proteinChemistrySuperoxideBiologyBiochemistryProtein kinase AKinaseEnzymeAdipose tissueBrown adipose tissueSulfur Compounds in BiologyEicosanoids and Hypertension PharmacologyRenin-Angiotensin System Studies
SQR mediates therapeutic effects of H <sub>2</sub> S by targeting mitochondrial electron transport to induce mitochondrial uncoupling | Litcius