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Extrahelical Binding Site for a 1H-Imidazo[4,5-c]quinolin-4-amine A3 Adenosine Receptor Positive Allosteric Modulator on Helix 8 and Distal Portions of Transmembrane Domains 1 and 7

Courtney Fisher, Matteo Pavan, Veronica Salmaso, Robert F. Keyes, Tina C. Wan, Balaram Pradhan, Zhan‐Guo Gao, Brian C. Smith, Kenneth A. Jacobson, John A. Auchampach

2024Molecular Pharmacology10 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryStereochemistryAllosteric regulationTransmembrane domainAmine gas treatingCrystallographyDocking (animal)Helix (gastropod)Molecular dynamicsBinding siteMolecular switchMoleculeAmino acidReceptorComputational chemistryBiochemistrySnailMedicineBiologyEcologyNursingOrganic chemistryReceptor Mechanisms and SignalingAdenosine and Purinergic SignalingPharmacological Receptor Mechanisms and Effects
Extrahelical Binding Site for a 1H-Imidazo[4,5-c]quinolin-4-amine A3 Adenosine Receptor Positive Allosteric Modulator on Helix 8 and Distal Portions of Transmembrane Domains 1 and 7 | Litcius