One molecule two goals: A selective P-glycoprotein modulator increases drug transport across gastro-intestinal barrier and recovers doxorubicin toxicity in multidrug resistant cancer cells
Marialessandra Contino, Stefano Guglielmo, Chiara Riganti, Giulia Antonello, Maria Grazia Perrone, Roberta Giampietro, Barbara Rolando, Roberta Fruttero, Nicola Antonio Colabufo
Topics & Concepts
ChemistryP-glycoproteinBioavailabilityToxicityPharmacologyDoxorubicinTransporterIn vitroEffluxATP-binding cassette transporterCaco-2Multiple drug resistanceBiochemistryChemotherapyBiologyGeneGeneticsAntibioticsOrganic chemistryDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesTrace Elements in Health