Discovery of 4-amino-1H-pyrazolo[3,4-d]pyrimidin derivatives as novel discoidin domain receptor 1 (DDR1) inhibitors
Ru Dong, Xin Zhou, Min Wang, Wen Li, Jinyang Zhang, Xin Xiao Zheng, Kai‐Xiang Tang, Li‐Ping Sun
Topics & Concepts
DDR1Discoidin domainChemistryReceptor tyrosine kinaseCell growthKinaseTyrosine kinasePlatelet-derived growth factor receptorIC50Cancer researchReceptorBiochemistryBiologyIn vitroGrowth factorCell Adhesion Molecules ResearchMonoclonal and Polyclonal Antibodies ResearchHER2/EGFR in Cancer Research