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Nickel-Catalyzed Homologation of Vinylidene Difluoride (CH<sub>2</sub>═CF<sub>2</sub>): Selective β-F <i>vs</i> β-H Elimination

Alexandre J. Sicard, Behnaz Ghaffari, Bulat Gabidullin, Jeffrey S. Ovens, Russell P. Hughes, R. Tom Baker

2022Journal of the American Chemical Society15 citationsDOI

Abstract

Hydrofluoroolefins (HFOs) constitute the newest generation of fluorocarbon refrigerants and foam-blowing agents due to their reduced global warming potential vs their saturated analogues. To identify new synthetic routes to HFOs, we show that reactions of bulky Ni(0) phosphine and −NHC complexes with vinylidene difluoride (VF2) afford μ-fluoro-1,1,3-trifluorobut-3-enyl Ni complexes. Moreover, addition of triisopropylsilane allows for reductive elimination of the reduced product─2,4,4-trifluoro-1-butene─demonstrating the Ni-catalyzed hydrodefluorodimerization of VF2. Accompanying DFT calculations identify the T-shaped nickelacyclopentane intermediate that spontaneously undergoes selective intramolecular β-F (vs β-H) elimination.

Topics & Concepts

ChemistryDifluorideCatalysisReductive eliminationPhosphineFluorocarbonNickelIntramolecular forceFluorideXenon difluorideMedicinal chemistryPolymer chemistryOrganic chemistryInorganic chemistryFluorine in Organic ChemistryInorganic Fluorides and Related CompoundsCarbon dioxide utilization in catalysis