Discovery of an Orally Available Diazabicyclooctane Inhibitor (ETX0282) of Class A, C, and D Serine β-Lactamases
Thomas F. Durand-Réville, Janelle Comita-Prevoir, Jing Zhang, Xiaoyun Wu, Tricia L. May‐Dracka, Jan Antoinette C. Romero, Frank Wu, April Chen, Adam B. Shapiro, Nicole Carter, Sarah M. McLeod, R.A. Giacobbe, Jeroen C. Verheijen, Sushmita D. Lahiri, M. Sacco, Yu Chen, John P. O’Donnell, Alita A. Miller, John P. Mueller, Rubén Tommasi
Abstract
infections.
Topics & Concepts
ChemistryProdrugAntibioticsPharmacologyOral administrationBioavailabilityEnzymeSerineBiochemistryMedicineAntibiotic Resistance in BacteriaAntibiotics Pharmacokinetics and EfficacyPneumocystis jirovecii pneumonia detection and treatment