Development of pyrazole and pyrazolopyrimidine derivatives as promising anti-MRSA agents targeting penicillin-binding protein (PBP2a) and mecA gene
Ahmed Ragab, Moustafa S. Abusaif, Heba Mohammed Refat M. Selim, Omnia Karem M. Riad, Mohamed H. Helal, Abeer M. Ali, Yousry A. Ammar, Ghada E. Ahmed
Topics & Concepts
ChemistryCandida albicansEscherichia coliPyrazoleADMEMicrobiologyAntibacterial activityStaphylococcus aureusBiofilmAntimicrobialGeneAntibioticsQuorum sensingBiochemistryBacteriaFluconazoleSCCmecMechanism of actionEffluxAntibacterial agentCorpus albicansVirulencePotencyBiological activityClick Chemistry and ApplicationsCancer therapeutics and mechanismsSynthesis and biological activity