New thieno[2,3-b]pyridine-fused pyrimidin-4(3H)-ones as potential thymidylate synthase inhibitors: Synthesis, SAR, in vitro and in silico study
Sherif M. H. Sanad, Ahmed E. M. Mekky
Topics & Concepts
ChemistryThymidylate synthaseCytotoxicityStereochemistryPyridineIn vitroBiochemistryMedicinal chemistryFluorouracilSurgeryMedicineChemotherapyBiochemical and Molecular ResearchCancer therapeutics and mechanismsSynthesis and biological activity