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Targeting platinum-resistant ovarian cancer by disrupting histone and RAD51 lactylation

Chenggong Sun, Xiao Li, Qiuli Teng, Xihan Liu, Li Song, Helgi B. Schiöth, Huan Wu, Xinyue Ma, Zhaoyang Zhang, Changjian Qi, H. C. Zhang, Kun Song, Qing Zhang, Beihua Kong

2025Theranostics56 citationsDOIOpen Access PDF

Abstract

Our study demonstrated the essential role of histone and RAD51 lactylation in HR repair and platinum resistance. It also identified a potential therapeutic strategy to overcome platinum resistance and improve prognosis in ovarian cancer.

Topics & Concepts

Ovarian cancerHistoneCancer researchRAD51PlatinumMedicineInternal medicineOncologyChemistryBiologyCancerBiochemistryDNA damageGeneDNACatalysisRNA modifications and cancerCancer-related molecular mechanisms researchMicroRNA in disease regulation
Targeting platinum-resistant ovarian cancer by disrupting histone and RAD51 lactylation | Litcius