EZH2 PROTACs target EZH2- and FOXM1-associated oncogenic nodes, suppressing breast cancer cell growth
Joshua M. Corbin, Xufen Yu, Jian Jin, Ling Cai, Gang Greg Wang
Topics & Concepts
EZH2FOXM1BiologyTamoxifenCancer researchPRC2Breast cancerHistone methyltransferaseTranscription factorMethylationCell cycleCancerGeneticsGeneProtein Degradation and InhibitorsHistone Deacetylase Inhibitors ResearchEpigenetics and DNA Methylation