Discovery of pomalidomide-based PROTACs for selective degradation of histone deacetylase 8
Zhiqiang Sun, Bulian Deng, Zichao Yang, Ruiyao Mai, Junli Huang, Zeli Ma, Ting Chen, Jianjun Chen
Topics & Concepts
HDAC8ChemistryHistone deacetylaseAcetylationUbiquitinHDAC6HDAC1BiochemistryProteolysisPomalidomideHistoneEnzymeBiologyBortezomibGeneMultiple myelomaImmunologyHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsPeptidase Inhibition and Analysis