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Discovery and structure-activity relationship studies of novel α-ketoamide derivatives targeting the SARS-CoV-2 main protease

Chong Huang, Rui Zeng, Jingxin Qiao, Baoxue Quan, Rong‐Hua Luo, Qiao Huang, Nihong Guo, Yueyue Li, Xin‐Yan Long, Ronggang Ma, Anjie Xia, Zhen Fang, Yifei Wang, Yueshan Li, Yong‐Tang Zheng, Linli Li, Jian Lei, Shengyong Yang, Jian Lei, Shengyong Yang

2023European Journal of Medicinal Chemistry15 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryProteasesProteaseDrug discoveryEnzymeStructure–activity relationshipIn vitroStereochemistryBiochemistrySARS-CoV-2 and COVID-19 ResearchComputational Drug Discovery MethodsViral Infections and Immunology Research
Discovery and structure-activity relationship studies of novel α-ketoamide derivatives targeting the SARS-CoV-2 main protease | Litcius