New potent ciprofloxacin-uracil conjugates as DNA gyrase and topoisomerase IV inhibitors against methicillin-resistant Staphylococcus aureus
Mohamed Samir, Mohamed Ramadan, Mostafa Abdelrahman, Mohammed A. I. Elbastawesy, Hamada Mohamed Halby, Mohamed Abdel‐Aziz, Gamal El‐Din A. Abuo‐Rahma
Topics & Concepts
DNA gyraseTopoisomerase IVCiprofloxacinChemistryTopoisomeraseStaphylococcus aureusAntibacterial activityIC50StereochemistryAntibacterial agentMinimum inhibitory concentrationDNAAntibioticsBiochemistryBacteriaIn vitroEscherichia coliBiologyGeneGeneticsCancer therapeutics and mechanismsAntibiotic Resistance in BacteriaAntibiotics Pharmacokinetics and Efficacy