Litcius/Paper detail

Current progress and novel strategies that target CDK12 for drug discovery

Peng Lei, Jifa Zhang, Pei‐Yu Liao, Changyu Ren, Jiaxing Wang, Di Wang

2022European Journal of Medicinal Chemistry22 citationsDOIOpen Access PDF

Topics & Concepts

Drug discoveryDNA damageDrug developmentDNA repairSynthetic lethalityBiologyComputational biologyCancer researchDrugChemistryBioinformaticsGeneticsDNAPharmacologyProtein Degradation and InhibitorsAdvanced Breast Cancer TherapiesUbiquitin and proteasome pathways