Litcius/Paper detail

Rescuing Tetracycline Class Antibiotics for the Treatment of Multidrug-Resistant Acinetobacter baumannii Pulmonary Infection

David M. P. De Oliveira, Brian M. Forde, Minh‐Duy Phan, Bernhard Steiner, Bing Zhang, Johannes Zuegg, Ibrahim M. El‐Deeb, Gen Li, Nadia Keller, Stephan Brouwer, Nichaela Harbison-Price, Amanda J. Cork, Michelle J. Bauer, Saleh F. Alquethamy, Scott A. Beatson, Jason A. Roberts, David L. Paterson, Alastair G. McEwan, Mark A. T. Blaskovich, Mark A. Schembri, Christopher A. McDevitt, Mark von Itzstein, Mark J. Walker

2022mBio26 citationsDOIOpen Access PDF

Abstract

Within intensive care unit settings, multidrug-resistant (MDR) Acinetobacter baumannii is a major cause of ventilator-associated pneumonia, and hospital-associated outbreaks are becoming increasingly widespread. Antibiotic treatment of A. baumannii infection is often compromised by MDR strains resistant to last-resort β-lactam (e.g., carbapenems), polymyxin, and tetracycline class antibiotics. During the on-going COVID-19 pandemic, secondary bacterial infection by A. baumannii has been associated with a 2-fold increase in COVID-19-related mortality. With a rise in antibiotic resistance and a reduction in new antibiotic discovery, it is imperative to investigate alternative therapeutic regimens that complement the use of current antibiotic treatment strategies. Rescuing the efficacy of existing therapies for the treatment of MDR A. baumannii infection represents a financially viable pathway, reducing time, cost, and risk associated with drug innovation.

Topics & Concepts

Acinetobacter baumanniiTigecyclineTetracyclineMicrobiologyMultiple drug resistanceAntibioticsPolymyxinMedicineAntibiotic resistanceColistinPneumoniaBiologyPseudomonas aeruginosaBacteriaInternal medicineGeneticsAntibiotic Resistance in BacteriaPneumonia and Respiratory InfectionsAntibiotics Pharmacokinetics and Efficacy