Development and application of novel electrophilic warheads in target identification and drug discovery
Yue Liu, Shumin Lv, Lijie Peng, Chengliang Xie, Liqian Gao, Hongyan Sun, Ligen Lin, Ke Ding, Zhengqiu Li
Topics & Concepts
DruggabilityDrug discoveryElectrophileWarheadComputational biologyAmino acidCombinatorial chemistryChemistryAmino acid residueDrug developmentBiochemistryDrugFunction (biology)BiologyPeptide sequencePharmacologyCell biologyCatalysisGeneEngineeringAerospace engineeringClick Chemistry and ApplicationsChemical Synthesis and AnalysisCannabis and Cannabinoid Research