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In silico, in vitro, and in vivo human metabolism of acetazolamide, a carbonic anhydrase inhibitor and common “diuretic and masking agent” in doping

Francesco Paolo Busardò, Alfredo Fabrizio Lo Faro, Ascanio Sirignano, Raffaele Giorgetti, Jérémy Carlier

2022Archives of Toxicology28 citationsDOI

Topics & Concepts

AcetazolamideChemistryMetaboliteIn vivoUrineGlucuronidationChromatographyCarbonic anhydraseMetabolismBiochemistryPharmacologyEnzymeInternal medicineMedicineMicrosomeBiologyBiotechnologyEnzyme function and inhibitionCholinesterase and Neurodegenerative DiseasesPharmacogenetics and Drug Metabolism
In silico, in vitro, and in vivo human metabolism of acetazolamide, a carbonic anhydrase inhibitor and common “diuretic and masking agent” in doping | Litcius