Synthesis, bioinformatics and biological evaluation of novel pyridine based on 8-hydroxyquinoline derivatives as antibacterial agents: DFT, molecular docking and ADME/T studies
Mohamed Rbaa, Asmaa Oubihi, Halima Hajji, Burak Tüzün, Abdelhadi Hichar, El Hassane Anouar, Elyor Berdimurodov, Mohammed Aziz Ajana, A. Zarrouk, B. Lakhrissi
Topics & Concepts
ChemistryADMECombinatorial chemistryDocking (animal)8-HydroxyquinolinePyridineAntibacterial activityComputational biologyBiochemistryOrganic chemistryBacteriaIn vitroMedicineGeneticsNursingBiologySynthesis and biological activityComputational Drug Discovery MethodsBioactive Compounds and Antitumor Agents