Design, synthesis and evaluation of novel indirubin-based N-hydroxybenzamides, N-hydroxypropenamides and N-hydroxyheptanamides as histone deacetylase inhibitors and antitumor agents
Duong Tien Anh, Hai Pham‐The, Đỗ Thị Mai Dung, Phan Thị Phương Dung, Huong Le‐Thi‐Thu, Eun Jae Park, Hye Won Jun, Jong Soon Kang, Joo‐Hee Kwon, Trương Thanh Tùng, Sang‐Bae Han, Nguyen‐Hai Nam
Topics & Concepts
ChemistryHistone deacetylaseIndirubinStereochemistryHistone deacetylase inhibitorChemical synthesisHistonePharmacologyCombinatorial chemistryBiochemistryIn vitroVisual artsIndigoMedicineArtGeneHistone Deacetylase Inhibitors ResearchQuinazolinone synthesis and applicationsClick Chemistry and Applications