Pharmacophore hybridization approach to discover novel pyrazoline-based hydantoin analogs with anti-tumor efficacy
Neha Upadhyay, Kalpana Tilekar, Fulvio Loiodice, N. Yu. Anisimova, Tatiana S. Spirina, Darina V. Sokolova, Galina B. Smirnova, Jun‐yong Choe, Franz‐Josef Meyer‐Almes, Vadim S. Pokrovsky, Antonio Lavecchia, C. S. Ramaa
Topics & Concepts
ChemistryHydantoinPyrrolidinePharmacophoreIn vivoPyrazolineStereochemistryIn vitroApoptosisPharmacologyCancer researchBiochemistryBiologyOrganic chemistryBiotechnologySynthesis and biological activitySynthesis of heterocyclic compoundsBioactive Compounds and Antitumor Agents